SCHEMBL9263229

SCHEMBL9263229

ClCc1nc(Cl)c2c(Cl)cccc2n1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.41
PARP1 P09874 2/20 0.40
GRIN1 Q05586 4/20 0.37
GRIN2A Q12879 4/20 0.37
ACHE P22303 3/20 0.37
ELANE P08246 3/20 0.37
BCHE P06276 2/20 0.36
DHFR P00374 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
PSMB8 P28062 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31663247 0.82 PARP1 (0.45) PARP1GRIN1GRIN2AACHEELANE
SCHEMBL3107616 0.82 KMT2A (0.39) KMT2APARP1ACHEELANEBCHE
SCHEMBL5234447 0.81 PARP1 (0.41) PARP1GRIN1GRIN2AACHEELANE
SCHEMBL9258621 0.78 GRIN1 (0.36) KMT2APARP1GRIN1GRIN2AACHE
SCHEMBL30013654 0.76 PARP1 (0.44) PARP1GRIN1GRIN2AACHEELANE
SCHEMBL3337344 0.76 PARP1 (0.44) PARP1GRIN1GRIN2AACHEELANE
SCHEMBL7417855 0.73 PARP1 (0.50) KMT2APARP1GRIN1GRIN2AACHE
SCHEMBL92745 0.73 KMT2A (0.50) KMT2AACHETDP1
SCHEMBL15537493 0.71 ALDH1A1 (0.37) KMT2A
SCHEMBL31140889 0.70 PARP1 (0.46) PARP1GRIN1GRIN2AACHEELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed
EP-0519307-A2 Tetracyclic Imidazodiazepines F. HOFFMANN-LA ROCHE AG (CH) 1992-12-23 EP disclosed