SCHEMBL9265461

SCHEMBL9265461

CC(=O)NC(Cc1n[nH]c2ccccc12)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.47
KDM4E B2RXH2 3/20 0.46
YTHDC1 Q96MU7 1/20 0.46
STAT3 P40763 1/20 0.46
HIF1A Q16665 1/20 0.46
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
FLT3 P36888 1/20 0.44
CCNA1 P78396 1/20 0.44
ACE P12821 3/20 0.44
MAPT P10636 1/20 0.43
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
IDO1 P14902 2/20 0.43
TDO2 P48775 1/20 0.43
EGFR P00533 1/20 0.42
SRC P12931 1/20 0.42
TACR1 P25103 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415396 0.78 ACE (0.45) ACE
SCHEMBL7409601 0.78 ACE (0.45) ACE
SCHEMBL7409605 0.78 ACE (0.45) ACE
SCHEMBL7412626 0.78 ACE (0.40) ALOX15KDM4EYTHDC1STAT3HIF1A
SCHEMBL7416939 0.76 KDM4E (0.55) KDM4EYTHDC1STAT3HIF1ACCNA2
SCHEMBL29353985 0.76 KDM4E (0.55) KDM4EYTHDC1STAT3HIF1ACCNA2
SCHEMBL1519993 0.76 KDM4E (0.55) KDM4EYTHDC1STAT3HIF1ACCNA2
SCHEMBL31646447 0.76 KDM4E (0.55) KDM4EYTHDC1STAT3HIF1ACCNA2
SCHEMBL31642427 0.76 KDM4E (0.55) KDM4EYTHDC1STAT3HIF1ACCNA2
SCHEMBL8197473 0.76 MMP9 (0.52) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5472978-A Tachykinin antagonists for treating pain, migraine and antiinflammatory agents MERCK SHARP & DOHME LTD. (GB) 1995-12-05 US disclosed
EP-0593559-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LTD. (GB) 1994-04-27 EP disclosed
WO-1993001169-A2 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO disclosed