SCHEMBL9269552

SCHEMBL9269552

Cc1ccc(N)cc1C=Cc1nc(C(C)C)cs1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.35
ALDH1A1 P00352 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
CASP1 P29466 2/20 0.32
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
CASP6 P55212 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9269544 1.00 ALB (0.35) ALBALDH1A1SMN1; SMN2CASP1NOS3
SCHEMBL9261501 0.85 ALB (0.35) ALBALDH1A1KDM4EPOLBCYP3A4
SCHEMBL9261513 0.85 ALB (0.35) ALBALDH1A1KDM4EPOLBCYP3A4
SCHEMBL9256170 0.79 ALDH1A1 (0.40) ALBALDH1A1SMN1; SMN2KDM4ECYP3A4
SCHEMBL9256181 0.79 ALDH1A1 (0.40) ALBALDH1A1SMN1; SMN2KDM4ECYP3A4
SCHEMBL9260315 0.77 ALB (0.49) ALBTSHR
SCHEMBL5777449 0.77 ALB (0.49) ALBTSHR
SCHEMBL27572318 0.71 ALB (0.39) ALB
SCHEMBL5779199 0.71 ALB (0.39) ALB
SCHEMBL5775269 0.70 ALB (0.42) ALBNOS3NOS1NOS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5399702-A Leukotriene antagonists; antiasthmatic, antiallergen, and antianaphylactic agents HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
EP-0577003-A1 Thiazolylvinylphenyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 1994-01-05 EP disclosed
US-5273986-A A substituted phenylalkyleneamidophenyleneethylene thiazole HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed