SCHEMBL9280647

SCHEMBL9280647

[CH2]CCNCc1ccc(-c2noc(C(Cc3ccc(C)c(C)c3)c3cccc(Cl)c3)n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.44
S1PR1 P21453 4/20 0.41
S1PR3 Q99500 4/20 0.40
S1PR4 O95977 1/20 0.40
S1PR5 Q9H228 1/20 0.40
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 2/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27920250 0.91 PTPN1 (0.44) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9913930 0.90 PTPN1 (0.44) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9103709 0.89 S1PR1 (0.55) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9103441 0.86 S1PR1 (0.57) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9103408 0.85 PTPN1 (0.48) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9101175 0.81 PTPN1 (0.45) PTPN1S1PR1S1PR3MAPTTP53
SCHEMBL27920426 0.81 PTPN1 (0.44) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL28807635 0.80 PTPN1 (0.48) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL9912337 0.79 PTPN1 (0.44) PTPN1S1PR1S1PR3S1PR4S1PR5
SCHEMBL15675888 0.79 PTPN1 (0.42) PTPN1S1PR1S1PR3S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646021-A1 OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P)RECEPTOR MODULATORS Allergan, Inc. (US) 2013-10-09 EP claimed
WO-2012074730-A1 OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P)RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 WO claimed
EP-2646021-B1 OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P)RECEPTOR MODULATORS ALLERGAN INC (US) 2014-11-05 EP disclosed
EP-2646021-A1 OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P)RECEPTOR MODULATORS Allergan, Inc. (US) 2013-10-09 EP disclosed
WO-2012074730-A1 OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P)RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 WO disclosed