SCHEMBL9280969

SCHEMBL9280969

CC(=O)C(Br)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.52
CES2 O00748 2/20 0.49
CES1 P23141 2/20 0.49
NR4A1 P22736 1/20 0.43
NR4A2 P43354 1/20 0.43
NR4A3 Q92570 1/20 0.43
PTPN1 P18031 1/20 0.43
ACP3 P15309 1/20 0.42
EPHX2 P34913 1/20 0.41
FFAR1 O14842 3/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
SRD5A2 P31213 1/20 0.40
PDPK1 O15530 1/20 0.40
CNR2 P34972 1/20 0.40
PDE2A O00408 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448575 0.82 GSK3B (0.53) GSK3BCES2CES1PTPN1ACP3
SCHEMBL839084 0.81 CES2 (0.53) GSK3BCES2CES1PTPN1ACP3
SCHEMBL15228996 0.81 CES2 (0.45) GSK3BCES2
SCHEMBL840763 0.80 GSK3B (0.47) GSK3BCES2CES1EPHX2AKR1C3
SCHEMBL330908 0.79 CES2 (0.53) CES2ACP3AKR1C3AKR1C2
SCHEMBL23182220 0.78 CES2 (0.50) GSK3BCES2CES1NR4A1NR4A2
SCHEMBL13170119 0.78 CES2 (0.65) GSK3BCES2CES1NR4A1NR4A2
SCHEMBL330957 0.78 HDAC3 (0.44) CES2CES1PTPN1
SCHEMBL17634288 0.78 GSK3B (0.45) GSK3BCES2CES1PTPN1ACP3
SCHEMBL17634101 0.78 NPSR1 (0.47) GSK3BCES2CES1PTPN1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197900-A1 INHIBITORS OF HIF PROLYL HYDROXYLASE Merck Sharp & Dohme Corp. (US) 2017-08-02 EP disclosed
WO-2016049099-A1 INHIBITORS OF HIF PROLYL HYDROXYLASE MERCK SHARP & DOHME CORP. (US) 2016-03-31 WO disclosed
US-5405860-A Fungicides BAYER AKTIENGESELLSCHAFT (DE) 1995-04-11 US disclosed
US-4912122-A Triazolyl alkanones or triazolyl-alkanols BAYER AKTIENGESELLSCHAFT (DE) 1990-03-27 US disclosed
US-4776877-A FUNGICIDES BAYER AKTIENGESELLSCHAFT (DE) 1988-10-11 US disclosed
US-4772623-A FUNGICIDES, MICROBIOCIDES, PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1988-09-20 US disclosed
US-4582843-A FUNGICIDES, MICROBIOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1986-04-15 US disclosed