SCHEMBL9282500

SCHEMBL9282500

COc1ccc(C(C)N2CCC(C(=O)c3nc4ccccc4n3CCCCn3cnnn3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.48
TACR2 P21452 1/20 0.48
TACR1 P25103 1/20 0.48
LMNA P02545 2/20 0.44
POLB P06746 2/20 0.44
OPRM1 P35372 1/20 0.41
TSPO P30536 2/20 0.40
REN P00797 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
KCNH2 Q12809 4/20 0.38
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260991 0.86 HRH1 (0.51) HRH1TACR2TACR1LMNAPOLB
SCHEMBL9282529 0.83 HRH1 (0.40) HRH1TACR2TACR1LMNAREN
SCHEMBL9282339 0.83 HRH1 (0.39) HRH1TACR2TACR1LMNAPOLB
SCHEMBL9268456 0.82 TACR2 (0.53) HRH1TACR2TACR1LMNAPOLB
SCHEMBL9282864 0.82 HRH1 (0.47) HRH1TACR2TACR1KCNH2ALDH1A1
SCHEMBL9284043 0.79 HRH1 (0.51) HRH1TACR2TACR1KCNH2
SCHEMBL9259123 0.77 TACR2 (0.45) HRH1TACR2TACR1LMNAPOLB
SCHEMBL9264749 0.72 HRH1 (0.41) HRH1TACR2TACR1KCNH2MAPK1
SCHEMBL9260984 0.71 HRH1 (0.70) HRH1TACR2TACR1LMNAPOLB
SCHEMBL9259114 0.70 HRH1 (0.73) HRH1TACR2TACR1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed