SCHEMBL9268456

SCHEMBL9268456

COc1ccc(C(C)N2CCC(C(=O)c3nc4ccccc4n3CC(=O)O)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.53
TACR1 P25103 1/20 0.53
HRH1 P35367 1/20 0.53
PTGDR2 Q9Y5Y4 3/20 0.48
LMNA P02545 4/20 0.45
MAPT P10636 3/20 0.45
TSHR P16473 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
OPRM1 P35372 1/20 0.44
POLB P06746 2/20 0.44
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 2/20 0.44
TSPO P30536 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260991 0.85 HRH1 (0.51) TACR2TACR1HRH1LMNAOPRM1
SCHEMBL9259123 0.83 TACR2 (0.45) TACR2TACR1HRH1LMNAMAPT
SCHEMBL9282500 0.82 HRH1 (0.48) TACR2TACR1HRH1LMNAMAPT
SCHEMBL9268450 0.82 TACR2 (0.77) TACR2TACR1HRH1PTGDR2LMNA
SCHEMBL9268866 0.80 HRH1 (0.43) TACR2TACR1HRH1PTGDR2MAPT
SCHEMBL9260978 0.78 KDM4E (0.50) TACR2TACR1HRH1PTGDR2ALDH1A1
SCHEMBL9268872 0.74 TACR2 (0.44) TACR2TACR1HRH1PTGDR2ALDH1A1
SCHEMBL9260920 0.74 KDM4E (0.50) PTGDR2ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9253881 0.74 HRH1 (0.58) TACR2TACR1HRH1KDM4E
SCHEMBL9259114 0.73 HRH1 (0.73) TACR2TACR1HRH1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed