SCHEMBL9282936

SCHEMBL9282936

CCCCCc1nn(C2CCNCC2)c2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.42
HRH1 P35367 1/20 0.42
ADRA1B P35368 1/20 0.42
ABCB1 P08183 1/20 0.40
CNR2 P34972 2/20 0.40
KHK P50053 5/20 0.39
TEAD1 P28347 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38
SLC6A4 P31645 1/20 0.38
NSD3 Q9BZ95 1/20 0.37
HTR6 P50406 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
BRD4 O60885 1/20 0.35
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12564065 0.76 ABCB1 (0.43) ABCB1NSD3HTR6PTGDR2ALDH1A1
SCHEMBL2851940 0.76 KHK (0.47) ABCB1KHKNSD3HTR6ALDH1A1
SCHEMBL24117847 0.75 PTGDR2 (0.40) ADRA1AHRH1ADRA1BKHKTEAD1
Hydrochloric Acid SCHEMBL1991841 0.75 ABCB1 (0.43) ABCB1NSD3HTR6PTGDR2ALDH1A1
Hydrochloric Acid SCHEMBL15658181 0.74 KHK (0.46) ABCB1KHKSLC6A4NSD3HTR6
SCHEMBL9284262 0.73 SLC6A4 (0.49) SLC6A4HTR6
SCHEMBL19501177 0.72 ADRA1A (0.45) ADRA1AHRH1ADRA1BCNR2ALDH1A1
SCHEMBL27540455 0.72 PDE4A (0.45) CNR2PTGDR2
SCHEMBL24289745 0.71 TEAD1 (0.41) CNR2TEAD1TEAD4TEAD2SLC6A4
SCHEMBL3049374 0.70 ADRA1A (0.49) ADRA1AHRH1ADRA1BCNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5393761-A Treatment of nervous system disorders H. LUNDBECK A/S (DK) 1995-02-28 US disclosed
EP-0470039-B1 Novel 3-arylindole and 3-arylindazole derivatives LUNDBECK & CO AS H (DK) 1994-12-07 EP disclosed
EP-0470039-A2 Novel 3-arylindole and 3-arylindazole derivatives H. LUNDBECK A/S (DK) 1992-02-05 EP disclosed