SCHEMBL9287299

SCHEMBL9287299

Cc1nc(N)nc(Cl)c1C(C)O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NR1I2 O75469 1/20 0.33
AHR P35869 1/20 0.33
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
IKBKB O14920 1/20 0.32
IKBKE Q14164 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.31
TLR8 Q9NR97 1/20 0.31
CHRM4 P08173 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3393860 0.87 ADORA2A (0.38) ADORA2AADORA1LMNA
SCHEMBL15434656 0.85 KDM4E (0.39) KDM4EALDH1A1LMNA
SCHEMBL8513097 0.83 ADORA2A (0.36) KDM4EADORA2AADORA1NPSR1NR1I2
SCHEMBL9203918 0.82 ADORA2A (0.35) KDM4EADORA2AADORA1NPSR1NR1I2
SCHEMBL6026297 0.79 KMT2A (0.36) KDM4EADORA2AADORA1ALDH1A1KMT2A
SCHEMBL9286811 0.77 NPSR1 (0.39) KDM4EADORA2AADORA1NPSR1ALDH1A1
SCHEMBL15504772 0.76 ADORA2A (0.32) ADORA2AADORA1
SCHEMBL13823338 0.74 NPSR1 (0.35) KDM4ENPSR1
SCHEMBL12495771 0.73 ADORA2A (0.40) KDM4EADORA2AADORA1
SCHEMBL15429583 0.73 ALDH1A1 (0.31) KDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071511-A1 BENZOXAZEPINES AS INHIBITORS OF MTOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed