SCHEMBL9289396

SCHEMBL9289396

CN1C=C(c2noc(C(OC3CCCCC3)c3cccc(Cl)c3)n2)C=CC1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
FAAH O00519 1/20 0.35
GCK P35557 2/20 0.33
BCHE P06276 1/20 0.33
GRM5 P41594 2/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9289400 0.79 DRD2 (0.35) DRD2DRD4DRD3FAAHGCK
SCHEMBL9106483 0.74 GCK (0.41) DRD2DRD4DRD3FAAHGCK
SCHEMBL1152072 0.60 DRD3 (0.78) DRD2DRD4DRD3
SCHEMBL9109208 0.58 GCK (0.41) GCK
SCHEMBL2719856 0.57 DRD3 (0.49) DRD2DRD4DRD3BCHEGAA
SCHEMBL9109153 0.57 GCK (0.41) GCK
SCHEMBL12064967 0.56 DRD3 (0.52) DRD2DRD4DRD3
Fumaric Acid SCHEMBL9356787 0.55 DRD3 (0.62) DRD2DRD4DRD3BCHE
SCHEMBL22637544 0.55 MAPT (0.53) GRM5
SCHEMBL16043113 0.55 MAPT (0.53) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646026-A1 NOVEL OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTOR MODULATORS Allergan, Inc. (US) 2013-10-09 EP claimed
WO-2012074718-A1 NOVEL OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 WO claimed
EP-2646026-A1 NOVEL OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTOR MODULATORS Allergan, Inc. (US) 2013-10-09 EP disclosed
WO-2012074718-A1 NOVEL OXADIAZOLE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE (S1P) RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 WO disclosed