SCHEMBL9290256

SCHEMBL9290256

Cc1cccc2cc(NC(=O)OC(C)(C)C)ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.56
CA1 P00915 1/20 0.56
CA9 Q16790 1/20 0.56
KAT6A Q92794 1/20 0.47
LCK P06239 3/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP17A1 P05093 1/20 0.42
BRD4 O60885 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
JAK2 O60674 1/20 0.41
NAMPT P43490 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MAP4K4 O95819 1/20 0.41
ACSS2 Q9NR19 1/20 0.41
SYK P43405 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1600933 0.86 HSD17B1 (0.51) CA12CA1CA9KAT6AHDAC3
SCHEMBL14503717 0.85 CA12 (0.49) CA12CA1CA9KAT6ALCK
SCHEMBL30070953 0.85 CA12 (0.49) CA12CA1CA9KAT6ALCK
SCHEMBL22804504 0.85 CA12 (0.49) CA12CA1CA9KAT6ALCK
SCHEMBL29953227 0.83 CA12 (0.50) CA12CA1CA9KAT6AHDAC3
SCHEMBL14503720 0.82 TTK (0.48) CA12CA1CA9KAT6AHDAC3
SCHEMBL20067498 0.82 CA12 (0.46) CA12CA1CA9KAT6AHDAC3
SCHEMBL30216106 0.81 KAT6A (0.60) CA12CA1CA9KAT6ACYP1A2
SCHEMBL3403454 0.81 KAT6A (0.60) CA12CA1CA9KAT6ACYP1A2
SCHEMBL29652239 0.80 KAT6A (0.47) CA12CA1CA9KAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670787-B1 CYTOKINE INHIBITORS ITHERX PHARMA INC (US) 2012-05-30 EP disclosed