SCHEMBL9291317

SCHEMBL9291317

COc1ccc(-c2ccc(C3CC[CH]CC3)cc2)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.38
TGFBR1 P36897 2/20 0.37
ACVR1 Q04771 2/20 0.37
KCNH2 Q12809 1/20 0.36
FPR2 P25090 4/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
KDM1A O60341 4/20 0.34
ALOX5AP P20292 2/20 0.34
FEN1 P39748 2/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
APP P05067 1/20 0.33
IL2 P60568 1/20 0.33
MAP4K1 Q92918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26802110 0.88 S1PR1 (0.47) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL19986374 0.87 S1PR1 (0.49) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL9291266 0.86 KDM1A (0.38) FPR2PDE4AKDM1ACYP3A4CYP2C9
SCHEMBL172438 0.86 ESR2 (0.42) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL12437068 0.84 ESR2 (0.41) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL18287662 0.84 KDM1A (0.38) S1PR1TGFBR1ACVR1KCNH2KDM1A
SCHEMBL18712356 0.83 CYP3A4 (0.48) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL9291443 0.83 FPR2 (0.37) FPR2PDE4AKDM1A
SCHEMBL17614852 0.82 FPR2 (0.37) S1PR1TGFBR1ACVR1KCNH2FPR2
SCHEMBL9291245 0.82 PDE4A (0.34) FPR2PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356563-A Two plate electrooptical cell HOFFMANN-LA ROCHE INC. (US) 1994-10-18 US disclosed
US-5244597-A Liquid crystalline mixtures having a chiral tilted smectic phase HOFFMANN-LA ROCHE INC. (US) 1993-09-14 US disclosed
EP-0343487-A1 Cyclohexyl esters of alpha-fluoro/carboxylic acids F. HOFFMANN-LA ROCHE AG (CH) 1989-11-29 EP disclosed