SCHEMBL9293122

SCHEMBL9293122

CC(C)(C)[Si](C)(C)Oc1ccc(-c2cc(F)cc(Br)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.43
PGR P06401 3/20 0.39
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA9 Q16790 4/20 0.38
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CYP17A1 P05093 1/20 0.33
CYP21A2 P08686 1/20 0.33
CYP11B1 P15538 1/20 0.33
APLNR P35414 2/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
ALPL P05186 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366758 0.82 PREP (0.50) PREPCA12CA1CA9CYP17A1
SCHEMBL12493503 0.80 CA12 (0.37) PREPCA12CA1CA9CHRNB4
SCHEMBL9293349 0.80 PGR (0.36) PREPPGRCHRNB4CHRNA3CYP17A1
SCHEMBL2607317 0.80 PREP (0.51) PREPCA12CA1CA9RAB9A
SCHEMBL23491348 0.80 PREP (0.57) PREPCA12CA1CA9ALOX5AP
SCHEMBL2548669 0.76 PREP (0.46) PREPCA12CA1CA9ALOX5AP
SCHEMBL9293373 0.75 SLC6A2 (0.43) PREPCA12CA1CA9NPC1
SCHEMBL614621 0.74 PREP (0.47) PREPCA12CA1CA9APLNR
SCHEMBL6763899 0.74 PREP (0.53) PREPCA12CA1CA9ALOX5AP
SCHEMBL20364924 0.73 PREP (0.55) PREPCA12CA1CA9NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350846-A Antibiotics MERCK & CO., INC. (US) 1994-09-27 US disclosed
US-5208329-A Antibacterial agents MERCK & CO., INC. (US) 1993-05-04 US disclosed
US-5182385-A Chemical intermediates for bactericides MERCK & CO., INC. (US) 1993-01-26 US disclosed
EP-0467434-A1 2-Biphenyl-carbapenem antibacterial agents MERCK & CO. INC. (US) 1992-01-22 EP disclosed
EP-0464900-A2 2-Biphenyl-carbapenems MERCK & CO. INC. (US) 1992-01-08 EP disclosed
US-5025006-A Carbapenicillin antibiotics MERCK & CO., INC. (US) 1991-06-18 US disclosed
US-5011832-A 2-biphenyl-carbapenem antibacterial agents MERCK & CO., INC. (US) 1991-04-30 US disclosed