SCHEMBL9293197

SCHEMBL9293197

CC(C)(C)[Si](C)(C)Oc1cccc(-c2cccc(Br)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 6/20 0.43
GABRB3 P28472 6/20 0.43
GABRA5 P31644 6/20 0.43
GABRA3 P34903 6/20 0.43
CA12 O43570 4/20 0.41
CA1 P00915 4/20 0.41
CA9 Q16790 4/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
MAPT P10636 3/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GABRA1 P14867 5/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL232409 0.90 CA12 (0.45) CA12CA1CA9RAB9AMAPT
SCHEMBL4576483 0.88 CA12 (0.44) CA12CA1CA9RAB9AMAPT
SCHEMBL7706827 0.82 CA1 (0.50) CA12CA1CA9SMN1; SMN2TP53
SCHEMBL30758292 0.81 ABL1 (0.56) CA12CA1CA9NPC1RAB9A
SCHEMBL6158612 0.80 HSP90AA1 (0.50) CA12CA1CA9ALDH1A1HSP90AA1
SCHEMBL9293373 0.79 SLC6A2 (0.43) CA12CA1CA9NPC1RAB9A
SCHEMBL18529823 0.77 MAOB (0.43) CA12CA1CA9NPC1RAB9A
SCHEMBL4576012 0.77 CA12 (0.37) CA12CA1CA9MAPTGAA
SCHEMBL8076860 0.77 CA12 (0.37) CA12CA1CA9MAPTGAA
SCHEMBL3182564 0.77 CA12 (0.46) CA12CA1CA9SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350846-A Antibiotics MERCK & CO., INC. (US) 1994-09-27 US disclosed
US-5208329-A Antibacterial agents MERCK & CO., INC. (US) 1993-05-04 US disclosed
US-5182385-A Chemical intermediates for bactericides MERCK & CO., INC. (US) 1993-01-26 US disclosed
EP-0467434-A1 2-Biphenyl-carbapenem antibacterial agents MERCK & CO. INC. (US) 1992-01-22 EP disclosed
EP-0464900-A2 2-Biphenyl-carbapenems MERCK & CO. INC. (US) 1992-01-08 EP disclosed
US-5025006-A Carbapenicillin antibiotics MERCK & CO., INC. (US) 1991-06-18 US disclosed
US-5011832-A 2-biphenyl-carbapenem antibacterial agents MERCK & CO., INC. (US) 1991-04-30 US disclosed