SCHEMBL232409

SCHEMBL232409

CC(C)(C)[Si](C)(C)Oc1cccc(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.45
CA1 P00915 4/20 0.45
CA9 Q16790 4/20 0.45
MAOB P27338 8/20 0.42
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EGFR P00533 2/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4576483 0.98 CA12 (0.44) CA12CA1CA9MAOBCYP1A2
SCHEMBL9293197 0.90 GABRG2 (0.43) CA12CA1CA9CYP1A2GAA
SCHEMBL7706827 0.88 CA1 (0.50) CA12CA1CA9CYP1A2GAA
SCHEMBL6158612 0.85 HSP90AA1 (0.50) CA12CA1CA9MAOBHSP90AA1
SCHEMBL9718082 0.84 MAOB (0.37) CA12CA1CA9MAOBCYP1A2
SCHEMBL4576012 0.83 CA12 (0.37) CA12CA1CA9MAOBCYP1A2
SCHEMBL18529823 0.83 MAOB (0.43) CA12CA1CA9MAOBCYP1A2
SCHEMBL8076860 0.83 CA12 (0.37) CA12CA1CA9CYP1A2GAA
SCHEMBL3182564 0.82 CA12 (0.46) CA12CA1CA9MAOBGAA
SCHEMBL3428405 0.82 MAOB (0.46) MAOBCYP1A2GAAMAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 277 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116041153-B Direct cross coupling method of aryl thioether and aryl bromine 南京工业大学 2024-05-24 CN claimed
CN-116253623-B Direct cross-coupling method of aryl fluorine sulfate and aryl bromine 南京工业大学 2024-04-05 CN claimed
CN-116554009-A Electrophilic cross-coupling reaction method of aryl sulfone or heteroaryl sulfone and aryl bromide 南京工业大学 2023-08-08 CN claimed
CN-116283515-A Direct cross coupling method of aryl fluoride and aryl bromide 南京工业大学 2023-06-23 CN claimed
CN-116253623-A Direct cross-coupling method of aryl fluorine sulfate and aryl bromine 南京工业大学 2023-06-13 CN claimed
CN-116041153-A Direct cross coupling method of aryl thioether and aryl bromine 南京工业大学 2023-05-02 CN claimed
US-20190010173-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS MATEON THERAPEUTICS, INC. (US) 2019-01-10 US claimed
WO-2017030983-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS MATEON THERAPEUTICS, INC. (US) 2017-02-23 WO claimed
CN-117659017-B TRPML1/2 modulator compound, pharmaceutical composition, preparation method and application thereof 北京华益健康药物研究中心 2026-05-15 CN disclosed
US-12435040-B2 1,3-substituted cyclobutyl derivatives and uses thereof BAUSCH + LOMB IRELAND LIMITED (IE) 2025-10-07 US disclosed
CN-115916763-B Antiviral 1, 3-dioxoindene compounds 诺华股份有限公司 2025-06-03 CN disclosed
US-20250090491-A1 ANTIVIRAL 1,3-DI-OXO-INDENE COMPOUNDS NOVARTIS AG (CH) 2025-03-20 US disclosed
US-20240308965-A1 1,3-SUBSTITUTED CYCLOBUTYL DERIVATIVES AND USES THEREOF JPMORGAN CHASE BANK, N.A., AS SUCCESSOR AGENT 2024-09-19 US disclosed
US-12083092-B2 Antiviral 1,3-di-oxo-indene compounds NOVARTIS AG (CH) 2024-09-10 US disclosed
EP-0649414-A1 OPIOID DIARYLMETHYLPIPERAZINES AND PIPERIDINES THE WELLCOME FOUNDATION LIMITED (GB) 1995-04-26 EP disclosed
WO-1995004051-A1 PIPERAZINE COMPOUNDS USED IN THERAPY THE WELLCOME FOUNDATION LIMITED (GB) 1995-02-09 WO disclosed
WO-1993015062-A1 OPIOID DIARYLMETHYLPIPERAZINES AND PIPERIDINES THE WELLCOME FOUNDATION LIMITED (GB) 1993-08-05 WO disclosed
US-4195178-A Methylenecyclopentane derivatives THE UPJOHN COMPANY (US) 1980-03-25 US disclosed
US-4181798-A Methylenecyclopentane derivatives THE UPJOHN COMPANY (US) 1980-01-01 US disclosed
US-4100192-A Inter-phenylene-PG amides THE UPJOHN COMPANY (US) 1978-07-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12435040-B2 1,3-substituted cyclobutyl derivatives and uses thereof TRPV1, TRPV3, TRPV2 CA12 2835/4885CA1 3007/4885CA9 2433/4885
US-20240308965-A1 1,3-SUBSTITUTED CYCLOBUTYL DERIVATIVES AND USES THEREOF TRPV1, TRPV3, TRPV2 CA12 2835/4885CA1 3007/4885CA9 2433/4885
US-20250090491-A1 ANTIVIRAL 1,3-DI-OXO-INDENE COMPOUNDS IRF3, EIF2AK2, MAVS CA12 3710/4885CA1 4762/4885CA9 2522/4885
US-20190010173-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF CATHEPSINS CTSS, CTSB, CTSK CA12 2529/4885CA1 1252/4885CA9 1557/4885
US-12083092-B2 Antiviral 1,3-di-oxo-indene compounds IRF3, EIF2AK2, MAVS CA12 3710/4885CA1 4762/4885CA9 2522/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.