SCHEMBL9299503

SCHEMBL9299503

C#CCN(Cc1cc2c(=O)n(COC(=O)C(C)(C)C)c(C)nc2cc1C)c1ccc(C(=O)O)cc1

nearest known ligand 0.44

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.44
DHFR P00374 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299312 0.92 TYMS (0.46) NAMPTDHFR
SCHEMBL9249466 0.92 NAMPT (0.47) NAMPTDHFR
SCHEMBL5734367 0.89
SCHEMBL9298837 0.89 NAMPT (0.43) NAMPT
SCHEMBL9246347 0.89 NAMPT (0.54) NAMPTDHFR
SCHEMBL9221939 0.87 HDAC1 (0.34)
SCHEMBL8488936 0.86 NAMPT (0.38) NAMPT
SCHEMBL9388379 0.86 NAMPT (0.40) NAMPT
SCHEMBL8487164 0.85
SCHEMBL8485192 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5280027-A Quinazoline containing compound IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-01-18 US disclosed
EP-0459730-A2 Anti-tumour compounds ZENECA LIMITED (GB) 1991-12-04 EP disclosed