SCHEMBL9300523

SCHEMBL9300523

CC1(C)C=C(n2ccc(C(CCCOCc3ccccc3)OCc3ccccc3)cc2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ABCB1 P08183 4/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
MCHR1 Q99705 6/20 0.33
KCNH2 Q12809 5/20 0.33
MAOB P27338 1/20 0.31
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300816 0.86 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DABCB1
SCHEMBL9300056 0.84 PDE4A (0.36) PDE4APDE4BPDE4CPDE4DMAOB
SCHEMBL9299446 0.83 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DABCB1
SCHEMBL9300169 0.83 PDE4A (0.39) PDE4APDE4BPDE4CPDE4DABCB1
SCHEMBL9299763 0.83 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DMCHR1
SCHEMBL9299999 0.79 PDE4A (0.40) PDE4APDE4BPDE4CPDE4D
SCHEMBL9299993 0.79 PDE4A (0.38) PDE4APDE4BPDE4CPDE4D
SCHEMBL9685249 0.78 PDE4A (0.37) PDE4APDE4BPDE4CPDE4D
SCHEMBL9301343 0.78 ABCB1 (0.47) ABCB1CYP3A4ALOX15
SCHEMBL9301353 0.78 ABCB1 (0.47) ABCB1CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296492-A Certain chroman derivatives useful for treating symptoms caused by contraction of smooth muscles, circulatory diseases or epilepsy NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1994-03-22 US disclosed
EP-0518342-A1 Chroman derivatives Nippon Kayaku Kabushiki Kaisha (JP) 1992-12-16 EP disclosed