SCHEMBL9300526

SCHEMBL9300526

Cl/C=C/C1CCC(c2ccc(-c3ccc(Br)cc3)cc2)CC1.N#Cc1ccc(-c2ccc(C3CCC(/C=C/Cl)CC3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.38
HRH3 Q9Y5N1 2/20 0.38
KCNH2 Q12809 1/20 0.38
MAOB P27338 3/20 0.36
MAOA P21397 1/20 0.36
P2RY14 Q15391 1/20 0.36
EGLN2 Q96KS0 1/20 0.36
PAX8 Q06710 1/20 0.34
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
HDAC2 Q92769 1/20 0.34
GRIA1 P42261 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA3 P42263 1/20 0.34
SCD5 Q86SK9 2/20 0.33
MMP3 P08254 1/20 0.33
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
PTK2 Q05397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963232 0.93 HRH3 (0.42) KDM1AHRH3KCNH2MAOBP2RY14
SCHEMBL8963220 0.93 HRH3 (0.42) KDM1AHRH3KCNH2MAOBP2RY14
SCHEMBL8963107 0.89 HDAC2 (0.40) KDM1AKCNH2MAOBMAOAP2RY14
SCHEMBL8962800 0.89 GRIA1 (0.39) HRH3KCNH2MAOBMAOAEGLN2
SCHEMBL8962812 0.89 GRIA1 (0.39) HRH3KCNH2MAOBMAOAEGLN2
SCHEMBL8963099 0.89 HDAC2 (0.40) KDM1AKCNH2MAOBMAOAP2RY14
SCHEMBL8963065 0.85 GRIA1 (0.37) HRH3KCNH2MAOBMAOAP2RY14
SCHEMBL9300179 0.84 HDAC2 (0.43) KDM1AKCNH2MAOBMAOAHDAC2
SCHEMBL8962820 0.84 HDAC2 (0.43) KDM1AKCNH2MAOBMAOAHDAC2
SCHEMBL9475718 0.82 HRH3 (0.42) KDM1AHRH3KCNH2MAOBP2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed