SCHEMBL9300671

SCHEMBL9300671

CCOC(=O)CCOCc1cc(N)cc(Nc2c3ccccc3nc3ccccc23)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 13/20 0.66
TOP2B Q02880 8/20 0.66
KDM4E B2RXH2 2/20 0.46
POLB P06746 2/20 0.46
GLA P06280 1/20 0.46
ABCB1 P08183 1/20 0.43
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
RAD52 P43351 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM1A O60341 1/20 0.42
SLC2A1 P11166 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300848 0.95 TOP2A (0.64) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9301391 0.94 TOP2A (0.63) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9300363 0.90 TOP2A (0.68) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9301899 0.88 TOP2A (0.67) TOP2ATOP2BKDM4EPOLBMAPT
SCHEMBL9300538 0.87 TOP2A (0.63) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9300912 0.87 TOP2A (0.53) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9301714 0.87 TOP2A (0.64) TOP2ATOP2BPOLBKMT2ARAD52
SCHEMBL9299722 0.84 TOP2A (0.64) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9300667 0.84 TOP2A (0.53) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL9300642 0.83 TOP2A (0.60) TOP2ATOP2BKDM4EPOLBGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354864-A Antitumor agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-11 US claimed