SCHEMBL9300864

SCHEMBL9300864

COC(=O)c1ccc(C)nc1OS(=O)(=O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
CFTR P13569 1/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13473869 0.85 TUBB4A (0.50) NPC1RAB9ACFTRTUBB4ATUBB
SCHEMBL1373668 0.78 TDP1 (0.58) RAB9ASMN1; SMN2TDP1MAPTL3MBTL1
SCHEMBL9612713 0.77 GAA (0.39) NPC1RAB9ASMN1; SMN2SDHBMAPT
SCHEMBL21001740 0.77 SOS1 (0.40) NPC1RAB9ASMN1; SMN2CASP3SENP8
SCHEMBL2027363 0.77 PDCD1 (0.52) PDCD1CD274NPC1RAB9ASMN1; SMN2
SCHEMBL15350245 0.76 CNR2 (0.45) PDCD1CD274NPC1RAB9ASMN1; SMN2
SCHEMBL31674204 0.75 KDM4E (0.42) RAB9ASMN1; SMN2TUBB4ATUBBTUBA3C
SCHEMBL1680551 0.75 KMT2A (0.38) NPC1SMN1; SMN2CFTRSDHBTDP1
SCHEMBL9909243 0.75 GAA (0.46) NPC1RAB9ASMN1; SMN2SDHBTDP1
SCHEMBL27002452 0.74 KDM4E (0.38) NPC1RAB9ASMN1; SMN2CASP3SENP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994009002-A1 2-(AZA-9-FLUORENONYL)CARBAPENEM ANTIBACTERIAL AGENTS MERCK & CO., INC. (US) 1994-04-28 WO disclosed
US-5294610-A Staphylococcus; side effect reduction MERCK & CO. INC. (US) 1994-03-15 US disclosed