SCHEMBL9301720

SCHEMBL9301720

CC(N)C(=O)OCCOCc1cc(N)cc(Nc2c3ccccc3nc3ccccc23)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 9/20 0.66
TOP2B Q02880 8/20 0.66
KDM1A O60341 2/20 0.42
HDAC3 O15379 3/20 0.41
HDAC4 P56524 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC7 Q8WUI4 3/20 0.41
HDAC2 Q92769 3/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC9 Q9UKV0 3/20 0.41
HDAC5 Q9UQL6 3/20 0.41
POLB P06746 3/20 0.41
RAD52 P43351 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MITF O75030 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301716 1.00 TOP2A (0.66) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL9301714 0.85 TOP2A (0.64) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL9301899 0.83 TOP2A (0.67) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL9300671 0.82 TOP2A (0.66) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL9300848 0.82 TOP2A (0.64) TOP2ATOP2BPOLBRAD52L3MBTL1
SCHEMBL9301113 0.81 TOP2A (0.69) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL8490361 0.81 TOP2A (0.80) TOP2ATOP2BKDM1AHDAC3HDAC4
SCHEMBL9299556 0.81 TOP2A (0.60) TOP2ATOP2BKDM1APOLBRAD52
SCHEMBL9301391 0.81 TOP2A (0.63) TOP2ATOP2BPOLBKDM4E
SCHEMBL9301299 0.81 TOP2A (0.62) TOP2ATOP2BKDM1APOLBRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354864-A Antitumor agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-11 US claimed
US-5354864-A Antitumor agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-11 US disclosed
WO-1993023049-A1 3-(9-ACRIDINYLAMINO)-5-HYDROXYMETHYLANILINE DERIVATIVES AS ANTICANCER AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1993-11-25 WO disclosed