SCHEMBL9301895

SCHEMBL9301895

CC1(C)CCSc2ccc(C#Cc3cnc(CCCCC(=O)O)nc3)cc21

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.59
CYP26A1 O43174 3/20 0.59
RARB P10826 13/20 0.55
RARG P13631 13/20 0.55
RARA P10276 12/20 0.55
KMT2A Q03164 1/20 0.55
RXRA P19793 2/20 0.39
CRABP2 P29373 1/20 0.38
FFAR1 O14842 4/20 0.34
CYP26B1 Q9NR63 1/20 0.34
SSTR5 P35346 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665899 0.88 RARB (0.62) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6665585 0.86 CYP3A4 (0.64) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9302221 0.85 CYP3A4 (0.43) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301902 0.85 CYP3A4 (0.53) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301486 0.83 RARB (0.56) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL22198842 0.82 CYP3A4 (0.70) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301731 0.80 CYP26A1 (0.41) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8671034 0.79 CYP3A4 (0.51) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL19342900 0.78 RARB (0.72) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL19342939 0.77 RARB (0.61) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed