SCHEMBL9301902

SCHEMBL9301902

CC1(C)CCSc2ccc(C#Cc3cnnc(CCCCC(=O)O)c3)cc21

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.53
CYP26A1 O43174 4/20 0.53
RARB P10826 14/20 0.51
RARG P13631 14/20 0.51
RARA P10276 12/20 0.51
KMT2A Q03164 1/20 0.49
RXRA P19793 2/20 0.37
CRABP2 P29373 1/20 0.36
CYP26B1 Q9NR63 2/20 0.32
SSTR5 P35346 1/20 0.32
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302103 0.89 RARB (0.56) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9302949 0.88 CYP3A4 (0.57) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9302619 0.86 CYP3A4 (0.39) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301895 0.85 CYP3A4 (0.59) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301486 0.84 RARB (0.56) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9303533 0.81 CYP26A1 (0.39) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9303234 0.80 RARB (0.61) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9303655 0.77 CYP3A4 (0.43) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301893 0.75 CYP3A4 (0.52) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6665585 0.75 CYP3A4 (0.64) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed