SCHEMBL9302956

SCHEMBL9302956

CSC1(SC)CCOc2ccc(C#Cc3cnnc(CC(=O)O)c3)cc21

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.34
CYP26B1 Q9NR63 1/20 0.34
AKR1B1 P15121 1/20 0.33
ACACB O00763 4/20 0.31
RARA P10276 2/20 0.31
RARB P10826 2/20 0.31
RARG P13631 2/20 0.31
CYP3A4 P08684 1/20 0.31
CRABP2 P29373 1/20 0.31
S1PR5 Q9H228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303247 0.88 CYP3A4 (0.35) RARARARBRARGCYP3A4
SCHEMBL9304352 0.87 CYP26A1 (0.46) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL9301245 0.85
SCHEMBL6666824 0.85 CYP26A1 (0.34) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL6664615 0.84 CYP3A4 (0.35) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL6665587 0.83 CYP26A1 (0.38) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL9302600 0.83 CYP26A1 (0.33) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL9302106 0.81 CYP3A4 (0.33) RARARARBRARGCYP3A4
SCHEMBL6670288 0.80 CYP26A1 (0.39) CYP26A1CYP26B1AKR1B1ACACBRARA
SCHEMBL6669241 0.78 PRSS1 (0.36) CYP26A1CYP26B1AKR1B1ACACBRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed