SCHEMBL9302106

SCHEMBL9302106

CCOC(=O)CCCCc1cc(C#Cc2ccc3c(c2)C(SC)(SC)CCO3)cnn1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
RARG P13631 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
TBXAS1 P24557 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302931 0.89 RARA (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL9303247 0.89 CYP3A4 (0.35) CYP3A4RARARARBRARGKMT2A
SCHEMBL9303658 0.88
SCHEMBL6664873 0.87 CYP3A4 (0.37) CYP3A4RARARARBRARGKMT2A
SCHEMBL9673782 0.86 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL6665905 0.86 CYP3A4 (0.37) CYP3A4RARARARBRARGKMT2A
SCHEMBL9303290 0.86 CYP3A4 (0.35) CYP3A4RARARARBRARGKMT2A
SCHEMBL9817856 0.86 CYP4Z1 (0.38) CYP4F2CYP4A11
SCHEMBL9817777 0.83 PPARA (0.35) KMT2ACYP4F2CYP4A11
SCHEMBL6671545 0.83 CYP3A4 (0.42) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed