SCHEMBL9304042

SCHEMBL9304042

COc1cccc(CCC(=O)NCCc2c[nH]c3ccccc23)c1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.67
ACHE P22303 2/20 0.65
MTNR1A P48039 4/20 0.62
MTNR1B P49286 2/20 0.62
CDK4 P11802 1/20 0.62
CCND1 P24385 1/20 0.62
MEN1 O00255 3/20 0.61
NPC1 O15118 1/20 0.61
POLB P06746 1/20 0.61
RAB9A P51151 1/20 0.61
BCHE P06276 1/20 0.59
GFER P55789 1/20 0.59
MAPT P10636 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852870 0.96 GFER (0.65) KMT2AACHEMTNR1AMTNR1BCDK4
SCHEMBL11483618 0.91 KMT2A (0.68) KMT2AACHEMTNR1AMTNR1BCDK4
SCHEMBL9302255 0.85 GFER (0.70) KMT2AMTNR1AMEN1GFER
SCHEMBL9117842 0.84 MEN1 (0.76) KMT2AMTNR1AMEN1NPC1RAB9A
SCHEMBL9304098 0.84 MEN1 (0.67) KMT2AMTNR1AMEN1GFER
SCHEMBL1520049 0.82 KMT2A (0.66) KMT2AACHECDK4CCND1MEN1
Hydrochloric Acid SCHEMBL11478621 0.82 KMT2A (0.83) KMT2AACHECDK4CCND1MEN1
SCHEMBL5871022 0.82 KMT2A (0.73) KMT2AACHECDK4CCND1MEN1
SCHEMBL7677886 0.82 MEN1 (0.84) KMT2AMTNR1AMEN1NPC1RAB9A
SCHEMBL21255779 0.81 KMT2A (0.69) KMT2AMTNR1AMEN1GFERMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283343-A Melatonin antagonists WHITBY RESEARCH, INC. (US) 1994-02-01 US disclosed
US-5093352-A Melatonin inhibitor, sleep, 2-aryl N-acetyl tryptamine WHITBY RESEARCH, INC. (US) 1992-03-03 US disclosed
EP-0375726-A4 MELATONIN ANALOGUES 1991-01-30 EP disclosed
EP-0375726-A1 MELATONIN ANALOGUES Whitby Research Incorporated (US) 1990-07-04 EP disclosed
WO-1989001472-A1 MELATONIN ANALOGUES NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-02-23 WO disclosed