SCHEMBL9305007

SCHEMBL9305007

CCCc1cc2[nH]c(S)nc2cc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
KDM4E B2RXH2 1/20 0.44
NPBWR1 P48145 2/20 0.42
PIM3 Q86V86 1/20 0.39
PGK1 P00558 1/20 0.37
ALDH1A1 P00352 2/20 0.37
RIPK1 Q13546 2/20 0.36
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
POLB P06746 2/20 0.35
RAB9A P51151 2/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 3/20 0.35
GALR2 O43603 1/20 0.35
MAPT P10636 3/20 0.35
KCNJ1 P48048 1/20 0.35
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305016 0.95 GAA (0.51) GAAKDM4ENPBWR1PIM3PGK1
SCHEMBL9305196 0.84 GAA (0.51) GAAKDM4ENPBWR1PIM3PGK1
SCHEMBL9305213 0.78 GAA (0.51) GAAKDM4ENPBWR1PIM3PGK1
SCHEMBL9307163 0.73 GAA (0.41) GAAKDM4EPIM3PGK1ALDH1A1
SCHEMBL9304375 0.73 ALDH1A1 (0.51) GAAKDM4ENPBWR1PIM3PGK1
SCHEMBL29250318 0.72 SNCA (0.44) KDM4EPIM3ALDH1A1POLBMAPT
SCHEMBL9306048 0.68 GAA (0.43) GAA
SCHEMBL9306173 0.68 ALDH1A1 (0.45) GAAPIM3PGK1ALDH1A1RIPK1
SCHEMBL9305210 0.68 ALDH1A1 (0.57) GAAKDM4EPIM3PGK1ALDH1A1
SCHEMBL5008296 0.66 GAA (0.66) GAAKDM4EALDH1A1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed