SCHEMBL9305528

SCHEMBL9305528

COc1ccc2nc(C(CC(=O)O)C(O)=S)oc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.44
NPC1 O15118 2/20 0.44
APP P05067 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LCK P06239 1/20 0.43
TLR4 O00206 1/20 0.42
XDH P47989 1/20 0.42
NLRP3 Q96P20 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.40
GLO1 Q04760 1/20 0.40
SLC16A3 O15427 1/20 0.40
CTSA P10619 5/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10892271 0.93 RAB9A (0.49) RAB9ANPC1KDM4EMEN1KMT2A
SCHEMBL9305516 0.90 TLR4 (0.44) RAB9ANPC1APPMEN1KMT2A
SCHEMBL8972643 0.88 TP53 (0.53) RAB9AAPPKDM4EMEN1KMT2A
SCHEMBL9305511 0.83 NPC1 (0.44) RAB9ANPC1APPMEN1KMT2A
SCHEMBL9305097 0.83 MAPT (0.49) RAB9ANPC1KDM4EMEN1KMT2A
SCHEMBL10892262 0.82 RAB9A (0.46) RAB9ANPC1KDM4EMEN1KMT2A
SCHEMBL8972467 0.82 MAPT (0.40) RAB9ANPC1KDM4EMEN1KMT2A
SCHEMBL9306816 0.82 PIK3CG (0.42) RAB9AXDHNLRP3MAPT
SCHEMBL10888980 0.82 MAPT (0.43) RAB9ANPC1MEN1KMT2ATP53
SCHEMBL9304726 0.81 CTSA (0.38) TP53MAPTCTSAHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
US-4612049-A BENZOTHI ZOLYL THIO-, BENZIMIDAZOLYLTHIO- OR BENZOXAZOLYLTHIO-SUBSTITUTED CARBOXY ACID CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed