SCHEMBL9305810

SCHEMBL9305810

CN(C)CCCn1nc(-c2ccc(Br)cc2)c2cnccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.49
PRKCG P05129 5/20 0.41
PRKCB P05771 5/20 0.41
PRKCA P17252 5/20 0.41
GSK3B P49841 5/20 0.41
KCNH2 Q12809 2/20 0.41
PRKCD Q05655 2/20 0.41
PRKCZ Q05513 1/20 0.41
RPS6KA5 O75582 1/20 0.38
KDM4C Q9H3R0 2/20 0.38
TDP2 O95551 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
LSS P48449 1/20 0.36
NAMPT P43490 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304434 0.93 CYP2D6 (0.42) CYP2D6PRKCGPRKCBPRKCAGSK3B
SCHEMBL8137068 0.88 CYP2D6 (0.49) CYP2D6PRKCGPRKCBPRKCAGSK3B
SCHEMBL9303584 0.88 CYP2D6 (0.57) CYP2D6PRKCGPRKCBPRKCAGSK3B
SCHEMBL9303541 0.88 CYP2D6 (0.47) CYP2D6PRKCGPRKCBPRKCAGSK3B
Hydrochloric Acid SCHEMBL8135773 0.86 CYP2D6 (0.56) CYP2D6PRKCGPRKCBPRKCAGSK3B
Hydrochloric Acid SCHEMBL9263878 0.86 CYP2D6 (0.46) CYP2D6PRKCGPRKCBPRKCAGSK3B
Hydrochloric Acid SCHEMBL8127101 0.86 CYP2D6 (0.46) CYP2D6PRKCGPRKCBPRKCAGSK3B
SCHEMBL9305096 0.84 KDM4E (0.38) RPS6KA5TDP1CYP1A2CYP3A4NAMPT
SCHEMBL8141249 0.83 NAMPT (0.38) CYP2D6CYP1A2CYP3A4NAMPTKDM4E
SCHEMBL9304696 0.82 CYP2D6 (0.52) CYP2D6PRKCGPRKCBPRKCAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed