SCHEMBL930737

SCHEMBL930737

NC1=NC(c2cccc(Br)c2)(c2ccnc(C3CC3)c2)c2nccnc21

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.45
KCNH2 Q12809 1/20 0.45
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
HDAC4 P56524 2/20 0.31
HDAC3 O15379 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931386 0.83 BACE1 (0.67) BACE1KCNH2
SCHEMBL931345 0.83 BACE1 (0.67) BACE1KCNH2
SCHEMBL930937 0.83 BACE1 (0.67) BACE1KCNH2
SCHEMBL931305 0.80 BACE1 (0.54) BACE1KCNH2
SCHEMBL2463625 0.78 BACE1 (0.72) BACE1KCNH2
SCHEMBL930773 0.75 BACE1 (0.39) BACE1KCNH2
SCHEMBL930770 0.75 BACE1 (0.39) BACE1KCNH2
SCHEMBL930702 0.74 BACE1 (0.33) BACE1KCNH2
SCHEMBL930738 0.74 BACE1 (0.33) BACE1KCNH2HDAC4
SCHEMBL932097 0.71 BACE1 (0.39) BACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed