SCHEMBL931386

SCHEMBL931386

NC1=N[C@@](c2cccc(-c3cncnc3)c2)(c2ccnc(C3CC3)c2)c2nccnc21

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.67
KCNH2 Q12809 13/20 0.67
BACE2 Q9Y5Z0 7/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL930937 1.00 BACE1 (0.67) BACE1KCNH2BACE2
SCHEMBL931345 1.00 BACE1 (0.67) BACE1KCNH2BACE2
SCHEMBL931305 0.89 BACE1 (0.54) BACE1KCNH2BACE2
SCHEMBL930737 0.83 BACE1 (0.45) BACE1KCNH2
SCHEMBL930574 0.82 BACE1 (0.58) BACE1KCNH2BACE2
SCHEMBL931248 0.82 BACE1 (0.53) BACE1KCNH2BACE2
SCHEMBL6885096 0.80 BACE1 (0.51) BACE1KCNH2BACE2
SCHEMBL2468765 0.80 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL6887116 0.77 BACE1 (0.50) BACE1KCNH2BACE2
SCHEMBL931362 0.77 BACE1 (0.61) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed