SCHEMBL930771

SCHEMBL930771

COc1c(C)cc([C@]2(c3cccc(Br)c3)NC(N)c3nccnc32)cc1C

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRND Q07001 1/20 0.32
BACE1 P56817 3/20 0.32
BACE2 Q9Y5Z0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932098 0.93
SCHEMBL931080 0.93
SCHEMBL931363 0.83 BACE1 (0.52) BACE1BACE2
SCHEMBL929365 0.82 BACE1 (0.39) BACE1BACE2
SCHEMBL931144 0.82 BACE1 (0.39) BACE1BACE2
SCHEMBL3359177 0.78 BACE1 (0.35) BACE1BACE2
SCHEMBL930705 0.78 DPP4 (0.32) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL3360854 0.78
SCHEMBL3359125 0.77
SCHEMBL931233 0.77 BACE1 (0.58) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed