SCHEMBL9308330

SCHEMBL9308330

CCOC(=O)c1ccc(C)nc1C(=O)OCC

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.53
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA7 P43166 2/20 0.49
CA9 Q16790 2/20 0.49
CA14 Q9ULX7 2/20 0.49
CYP1A2 P05177 2/20 0.49
ALDH1A1 P00352 4/20 0.46
HSD17B10 Q99714 1/20 0.46
KDM4E B2RXH2 3/20 0.44
TARBP2 Q15633 1/20 0.44
CDC25B P30305 2/20 0.43
CDC25A P30304 1/20 0.43
CDC25C P30307 1/20 0.43
PDE4A P27815 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9355979 0.84 TSHR (0.55) TSHRMEN1KMT2ACA12CA1
SCHEMBL5664007 0.84 KDM4E (0.57) TSHRMEN1KMT2ACA12CA1
SCHEMBL13406205 0.84 KDM4E (0.50) TSHRMEN1KMT2ACA12CA1
SCHEMBL6306356 0.83 TSHR (0.50) TSHRMEN1KMT2ACA12CA1
SCHEMBL9308690 0.83 TSHR (0.50) TSHRMEN1KMT2ACA12CA1
SCHEMBL16828808 0.82 MEN1 (0.55) TSHRMEN1KMT2ACA12CA1
SCHEMBL7354531 0.82 TSHR (0.53) TSHRMEN1KMT2ACA12CA1
SCHEMBL6896843 0.81 ALDH1A1 (0.49) TSHRMEN1KMT2ACYP1A2ALDH1A1
SCHEMBL510572 0.81 ALDH1A1 (0.54) TSHRMEN1KMT2ACA12CA1
SCHEMBL4908919 0.81 TARBP2 (0.48) TSHRMEN1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5322948-A Reacting unsaturated diacid or derivative with hydroxylamine or a salt thereof to form N-hydroxy-2-aminobutane diacid derivative HOECHST CELANESE CORPORATION (US) 1994-06-21 US claimed
EP-0511446-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1992-11-04 EP claimed
EP-0456504-A2 Process for preparing pyridinecarboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-11-13 EP claimed
US-5047542-A Reaction of ketoester with unsaturated aldehyde or ketone HOECHST CELANESE CORPORATION (US) 1991-09-10 US claimed
EP-0415767-A2 Process for preparing pyridine carboxylic acid derivatives HOECHST CELANESE CORPORATION (US) 1991-03-06 EP claimed
US-4871859-A REACTING KETOESTER WITH UNSATURATED ALDEHYDE OR KETONE AND AMMONIUM SALT IN SOLVENT AND DEHYDROGENATION CATALYST HOECHST CELANESE CORPORATION 1989-10-03 US claimed
WO-1989008103-A1 PROCESS FOR PREPARING PYRIDINE CARBOXYLIC ACID ESTERS HOECHST CELANESE CORPORATION (US) 1989-09-08 WO claimed