SCHEMBL9309318

SCHEMBL9309318

Cc1ccc2c(-c3c(Br)cccc3C#N)occ2c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.33
MAOB P27338 2/20 0.32
MAOA P21397 1/20 0.32
DYRK1A Q13627 1/20 0.32
KDM4E B2RXH2 4/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
NPSR1 Q6W5P4 2/20 0.30
GAA P10253 2/20 0.30
RXFP1 Q9HBX9 1/20 0.30
PKM P14618 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550394 0.79 TSHR (0.36) CYP1A2KDM4EALDH1A1HPGDTSHR
SCHEMBL9309312 0.73 MAOB (0.57) MAOBMAOAALDH1A1
SCHEMBL9226415 0.69 CYP1A2 (0.57) CYP1A2KDM4EALDH1A1HPGDTSHR
SCHEMBL7822962 0.63 CYP1A2 (0.63) CYP1A2MAOBMAOAKDM4EALDH1A1
SCHEMBL29038987 0.63 CYP1A2 (0.49) CYP1A2MAOBMAOADYRK1AKDM4E
SCHEMBL15704191 0.63 CYP1A2 (0.57) CYP1A2MAOAKDM4EALDH1A1HPGD
SCHEMBL26794228 0.62 TSHR (0.38) CYP1A2DYRK1AKDM4ETSHRNPSR1
SCHEMBL1232348 0.61 TSHR (0.48) DYRK1AKDM4EALDH1A1TSHRLMNA
SCHEMBL306406 0.61 AR (0.42) MAOBMAOAALDH1A1HPGDTSHR
SCHEMBL8404426 0.61 CYP1A2 (0.46) CYP1A2MAOBKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5374646-A Treatment or prophylasix of hypertension and diseases associated with cognitive disorders GLAXO GROUP LIMITED (GB) 1994-12-20 US disclosed
CN-1052672-A Benzofuran derivative GLAXO GROUP LTD (GB) 1991-07-03 CN disclosed
EP-0434249-A2 Benzofuran derivatives GLAXO GROUP LIMITED (GB) 1991-06-26 EP disclosed