SCHEMBL9310028

SCHEMBL9310028

O=C(CCCN1CCC2c3ccccc3CCC2C1)c1ccc(F)cc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.62
HTR2C P28335 4/20 0.62
CCR3 P51677 1/20 0.62
SIGMAR1 Q99720 6/20 0.61
DRD3 P35462 2/20 0.61
HTR1A P08908 2/20 0.60
DRD4 P21917 1/20 0.60
SLC6A4 P31645 1/20 0.60
DRD2 P14416 2/20 0.57
HTR7 P34969 1/20 0.57
HRH1 P35367 1/20 0.57
HTR2B P41595 1/20 0.57
KDM4E B2RXH2 1/20 0.56
HSD17B10 Q99714 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8183381 0.77 DRD3 (0.65) HTR2ADRD3HTR1ADRD4DRD2
SCHEMBL5405231 0.77 HTR2A (1.00) HTR2AHTR2CCCR3HTR1ADRD4
SCHEMBL5847647 0.77 HTR2A (1.00) HTR2AHTR2CCCR3HTR1ADRD4
SCHEMBL9307016 0.77 SIGMAR1 (1.00) SIGMAR1
SCHEMBL9307027 0.77 SIGMAR1 (1.00) SIGMAR1
SCHEMBL9307633 0.77 SIGMAR1 (1.00) SIGMAR1
SCHEMBL9307021 0.77 SIGMAR1 (1.00) SIGMAR1
SCHEMBL11856580 0.76 HTR2A (0.69) HTR2AHTR2CCCR3HTR1ADRD4
SCHEMBL13904324 0.76 HTR2A (0.64) HTR2AHTR2CCCR3HTR1ADRD4
Hydrochloric Acid SCHEMBL9308495 0.76 SIGMAR1 (1.00) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5294618-A Psychological disorders MERCK SHARP & DOHME LIMITED (GB) 1994-03-15 US disclosed
EP-0410535-A2 Octahydrobenzisoquinoline derivatives as antipsychotic agents MERCK SHARP & DOHME LTD. (GB) 1991-01-30 EP disclosed