SCHEMBL9313974

SCHEMBL9313974

Cc1c(C)c2c(c(C)c1O)CCC(C)(CNc1ccccc1)O2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
TSHR P16473 2/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
CYP1A2 P05177 1/20 0.49
MAPT P10636 3/20 0.48
LMNA P02545 3/20 0.48
USP2 O75604 2/20 0.48
CYP2C9 P11712 2/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
GSTP1 P09211 1/20 0.48
TTPA P49638 1/20 0.48
THRB P10828 1/20 0.48
CYP2C19 P33261 1/20 0.48
ALOX5 P09917 5/20 0.48
CYP4F2 P78329 1/20 0.47
NR1I2 O75469 2/20 0.47
TP53 P04637 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690256 0.88 CYP4F2 (0.53) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9690390 0.82 ALOX5 (0.50) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9313902 0.81 BCHE (0.53) CYP3A4TSHRMAPTLMNAUSP2
SCHEMBL9689563 0.81 ALOX5 (0.49) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL18933886 0.80 MAPT (0.55) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL17289289 0.80 NR1I2 (0.50) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL20764885 0.80 NR1I2 (0.50) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9689071 0.80 ALOX5 (0.48) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9314063 0.80 MAPT (0.47) CYP3A4TSHRPTGS1PTGS2CYP1A2
SCHEMBL9689540 0.80 CYP4F2 (0.46) CYP3A4TSHRPTGS1PTGS2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP claimed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP claimed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP claimed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO claimed
US-5315017-A Peroxidation and eicosanoid biosynthesis inhibition ADIR ET COMPAGNIE (FR) 1994-05-24 US disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed