SCHEMBL931427

SCHEMBL931427

CC1=NC(CC2CCOCC2)(c2cccc(-c3cncc(F)c3)c2)N=C1N

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.49
KCNH2 Q12809 6/20 0.49
BACE2 Q9Y5Z0 3/20 0.49
APP P05067 1/20 0.43
GSK3B P49841 1/20 0.40
DYRK1A Q13627 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL943862 0.89 BACE1 (0.63) BACE1KCNH2BACE2APP
SCHEMBL932718 0.87 BACE1 (0.58) BACE1KCNH2BACE2
SCHEMBL932037 0.81 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL932274 0.78 BACE1 (0.43) BACE1KCNH2BACE2APP
SCHEMBL1076369 0.78 BACE1 (0.51) BACE1KCNH2BACE2APP
SCHEMBL931841 0.75 BACE1 (0.70) BACE1KCNH2BACE2APP
SCHEMBL932157 0.72 BACE1 (0.51) BACE1KCNH2BACE2
SCHEMBL932355 0.72 BACE1 (0.59) BACE1KCNH2BACE2APP
SCHEMBL932095 0.67 BACE1 (0.78) BACE1KCNH2BACE2
SCHEMBL1076368 0.67 BACE1 (0.43) BACE1KCNH2BACE2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed