SCHEMBL1076368

SCHEMBL1076368

COc1c(-c2ccccc2)cccc1C1(CC2CCOCC2)N=C(C)C(N)=N1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.43
KCNH2 Q12809 2/20 0.43
NPSR1 Q6W5P4 5/20 0.37
APP P05067 6/20 0.35
CTSD P07339 1/20 0.32
CTSE P14091 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075786 0.82 BACE1 (0.58) BACE1KCNH2APPBACE2
SCHEMBL1076369 0.79 BACE1 (0.51) BACE1KCNH2NPSR1APPBACE2
SCHEMBL932037 0.75 BACE1 (0.68) BACE1KCNH2BACE2
SCHEMBL946110 0.73 BACE1 (0.50) BACE1KCNH2APPBACE2
SCHEMBL946601 0.71 BACE1 (0.44) BACE1KCNH2
SCHEMBL932718 0.71 BACE1 (0.58) BACE1KCNH2CTSDBACE2
SCHEMBL932274 0.69 BACE1 (0.43) BACE1KCNH2NPSR1APPBACE2
SCHEMBL943862 0.67 BACE1 (0.63) BACE1KCNH2APPBACE2
SCHEMBL1076367 0.66 ALDH1A1 (0.33)
SCHEMBL1075789 0.65 BACE1 (0.74) BACE1KCNH2APPBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed