SCHEMBL9317686

SCHEMBL9317686

CC(=O)NCC(CCOS(C)(=O)=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.39
CYP2D6 P10635 4/20 0.39
SLC6A2 P23975 4/20 0.39
SLC6A4 P31645 4/20 0.39
SLC6A3 Q01959 4/20 0.39
KCNH2 Q12809 2/20 0.39
LMNA P02545 3/20 0.38
HTT P42858 2/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MCHR1 Q99705 4/20 0.37
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8118533 0.91 MCHR1 (0.39) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL8590813 0.85 S1PR3 (0.37) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL8782261 0.85 POLB (0.44) CYP2D6ALDH1A1HPGD
SCHEMBL8838875 0.79 CCKAR (0.39) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL9317560 0.79 TRPV1 (0.44) ALDH1A1MCHR1
SCHEMBL9318213 0.79 TACR2 (0.47)
SCHEMBL8835963 0.77 FNTA (0.49) CYP3A4SLC6A2LMNAHTT
SCHEMBL7809587 0.77 FNTA (0.53) LMNAALDH1A1HPGD
SCHEMBL7802907 0.73 ALDH1A1 (0.44) CYP3A4CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL4984205 0.73 TACR2 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350852-A Neurokinin A receptor antagonist SANOFI (FR) 1994-09-27 US disclosed
US-5236921-A Administrering for treatment of neutrogenic inflammation of the respiratory trart SANOFI (FR) 1993-08-17 US disclosed