SCHEMBL932046

SCHEMBL932046

CC1=NC(c2ccccc2)(c2cccc(Br)c2)N=C1N

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.60
KCNH2 Q12809 3/20 0.47
BACE2 Q9Y5Z0 1/20 0.44
APP P05067 3/20 0.41
CTSD P07339 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932108 0.90 BACE1 (0.62) BACE1KCNH2BACE2APPCTSD
SCHEMBL933512 0.89 BACE1 (0.63) BACE1KCNH2BACE2APPCTSD
SCHEMBL932111 0.87 BACE1 (0.47) BACE1KCNH2BACE2APPCTSD
SCHEMBL932706 0.86 BACE1 (0.66) BACE1KCNH2BACE2APPCTSD
SCHEMBL932757 0.84 BACE1 (0.44) BACE1KCNH2BACE2APPCTSD
SCHEMBL932204 0.83 BACE1 (0.67) BACE1KCNH2BACE2APP
SCHEMBL932844 0.82 BACE1 (0.50) BACE1KCNH2BACE2CTSD
SCHEMBL932806 0.82 BACE1 (0.41) BACE1KCNH2CTSD
SCHEMBL932503 0.82 BACE1 (0.67) BACE1KCNH2BACE2CTSD
SCHEMBL946979 0.81 BACE1 (0.42) BACE1KCNH2BACE2APPCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed