SCHEMBL932844

SCHEMBL932844

CC1=NC(c2ccc(OC(F)F)cc2)(c2cccc(Br)c2)N=C1N

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.50
KCNH2 Q12809 2/20 0.49
BACE2 Q9Y5Z0 4/20 0.41
REN P00797 3/20 0.41
CTSD P07339 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932551 0.86 BACE1 (0.40) BACE1KCNH2BACE2RENCTSD
SCHEMBL932706 0.85 BACE1 (0.66) BACE1KCNH2BACE2CTSD
SCHEMBL932215 0.85 BACE1 (0.41) BACE1KCNH2BACE2RENCTSD
SCHEMBL932175 0.85 BACE1 (0.51) BACE1KCNH2BACE2CTSD
SCHEMBL933512 0.83 BACE1 (0.63) BACE1KCNH2BACE2CTSD
SCHEMBL932046 0.82 BACE1 (0.60) BACE1KCNH2BACE2CTSD
SCHEMBL932390 0.81 BACE1 (0.77) BACE1KCNH2BACE2
SCHEMBL932108 0.79 BACE1 (0.62) BACE1KCNH2BACE2CTSD
SCHEMBL932111 0.76 BACE1 (0.47) BACE1KCNH2BACE2CTSD
SCHEMBL932503 0.76 BACE1 (0.67) BACE1KCNH2BACE2RENCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed