SCHEMBL932165

SCHEMBL932165

CC#Cc1cncc(-c2cc(C3(C4CC4)N=C(C)C(N)=N3)ccc2F)c1

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.79
KCNH2 Q12809 4/20 0.79
BACE2 Q9Y5Z0 4/20 0.71
APP P05067 10/20 0.48
CTSD P07339 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931947 0.89 BACE1 (1.00) BACE1KCNH2BACE2APPCTSD
SCHEMBL931695 0.85 BACE1 (0.70) BACE1KCNH2BACE2APP
SCHEMBL942561 0.84 BACE1 (0.57) BACE1KCNH2BACE2APPCTSD
SCHEMBL932246 0.83 BACE1 (1.00) BACE1KCNH2BACE2APPCTSD
SCHEMBL1032043 0.80 BACE1 (0.92) BACE1KCNH2BACE2APPCTSD
SCHEMBL21307771 0.75 BACE1 (0.68) BACE1KCNH2BACE2APPCTSD
SCHEMBL18562653 0.75 BACE1 (0.68) BACE1KCNH2BACE2APPCTSD
SCHEMBL6891149 0.74 BACE1 (0.58) BACE1KCNH2BACE2APP
SCHEMBL18561562 0.73 BACE1 (0.65) BACE1KCNH2BACE2APPCTSD
SCHEMBL18561441 0.73 BACE1 (0.65) BACE1KCNH2BACE2APPCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO claimed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed