SCHEMBL932350

SCHEMBL932350

COc1ccc(C2(c3cccc(Br)c3)N=C(N)C(S)=N2)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 17/20 0.50
KCNH2 Q12809 5/20 0.49
CTSD P07339 2/20 0.40
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
BACE2 Q9Y5Z0 2/20 0.36
RXFP1 Q9HBX9 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932706 0.86 BACE1 (0.66) BACE1KCNH2CTSDADORA2AADORA1
SCHEMBL932551 0.84 BACE1 (0.40) BACE1KCNH2CTSDBACE2
SCHEMBL932144 0.83 BACE1 (0.46) BACE1KCNH2CTSD
SCHEMBL932682 0.83 BACE1 (0.53) BACE1KCNH2CTSDBACE2
SCHEMBL932184 0.83 BACE1 (0.48) BACE1KCNH2CTSDADORA2AADORA1
SCHEMBL933481 0.77 BACE1 (0.39) BACE1KCNH2CTSDBACE2ALDH1A1
SCHEMBL932676 0.76 MAPT (0.38) BACE1CTSDBACE2ALDH1A1
SCHEMBL6922254 0.73 BACE1 (0.69) BACE1KCNH2CTSDBACE2
SCHEMBL932572 0.73 BACE1 (0.69) BACE1KCNH2CTSDBACE2
SCHEMBL932844 0.72 BACE1 (0.50) BACE1KCNH2CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed