SCHEMBL932602

SCHEMBL932602

COc1ccc(C2(c3cccc(Cl)c3)N=C(C)C(N)=N2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.56
KCNH2 Q12809 4/20 0.49
BACE2 Q9Y5Z0 2/20 0.47
FYN P06241 1/20 0.39
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DHPS P49366 1/20 0.37
CTSD P07339 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931620 0.86 BACE1 (0.43) BACE1KCNH2BACE2FYNMAPT
SCHEMBL932603 0.84 BACE1 (0.41) BACE1KCNH2BACE2FYNMAPT
SCHEMBL932404 0.80 BACE1 (0.86) BACE1KCNH2BACE2CTSD
SCHEMBL943241 0.74 BACE1 (0.46) BACE1KCNH2BACE2CTSD
SCHEMBL931686 0.74 BACE1 (0.53) BACE1KCNH2BACE2MAPTCTSD
SCHEMBL931578 0.73 BACE1 (0.45) BACE1KCNH2BACE2CTSD
SCHEMBL932572 0.73 BACE1 (0.69) BACE1KCNH2BACE2CTSD
SCHEMBL6922254 0.73 BACE1 (0.69) BACE1KCNH2BACE2CTSD
SCHEMBL943682 0.71 BACE1 (0.47) BACE1KCNH2BACE2CTSD
SCHEMBL932245 0.70 BACE1 (0.79) BACE1KCNH2BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002407-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed