SCHEMBL9326541

SCHEMBL9326541

O=C(O)Cc1ccc2c(c1)CNC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
MAPT P10636 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
ALDH1A1 P00352 3/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
GAA P10253 4/20 0.48
TSHR P16473 3/20 0.48
LMNA P02545 2/20 0.48
NFKB1 P19838 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
RGS12 O14924 1/20 0.48
POLB P06746 1/20 0.48
APEX1 P27695 1/20 0.48
THPO P40225 1/20 0.48
BLM P54132 1/20 0.48
GNAI1 P63096 1/20 0.48
PMP22 Q01453 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27919835 0.98 KDM4E (0.47) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL31478167 0.79 AKR1B1 (0.58) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL26133994 0.77 ITGB3 (0.45) KDM4EMAPTALDH1A1TSHRPOLB
SCHEMBL3838996 0.77 RXRB (0.62) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL1206291 0.76 HTR2A (0.40) ITGB3ITGA2B
SCHEMBL31514914 0.76 HTR2A (0.40) ITGB3ITGA2B
SCHEMBL5527444 0.76 RXRB (0.65) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL19996854 0.76 RXRB (0.60) KDM4EMAPTHPGDHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL3710885 0.75 HTR2A (0.39) ITGB3ITGA2B
SCHEMBL5173443 0.74 GAA (0.48) KDM4EMAPTHPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3166925-A1 ISOINDOLINE DERIVATIVES FOR USE IN THE TREATMENT OF A VIRAL INFECTION VIIV Healthcare UK Limited (GB) 2017-05-17 EP disclosed
WO-2016005878-A1 ISOINDOLINE DERIVATIVES FOR USE IN THE TREATMENT OF A VIRAL INFECTION VIIV HEALTHCARE UK LIMITED (GB) 2016-01-14 WO disclosed
CN-104045552-A Medicinal compound as neuroprotective agent SHANGHAI SIMCERE PHARMACEUTICAL RES CO LTD 2014-09-17 CN disclosed
CN-103313968-A Nampt and rock inhibitors ABBVIE LAB 2013-09-18 CN disclosed
US-5288749-A Treating central nervous system or cardiovascular disorders ABBOTT LABORATORIES (US) 1994-02-22 US disclosed