SCHEMBL9326962

SCHEMBL9326962

Nc1nc(NC2CCCC2)nc2nc(-c3ccco3)nn12

nearest known ligand 0.98

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.98
ADORA1 P30542 13/20 0.98
ADORA3 P0DMS8 12/20 0.98
ADORA2B P29275 3/20 0.98
CSNK1D P48730 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9327282 0.99 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BCSNK1D
SCHEMBL5408777 0.84 ADORA2A (0.71) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9325961 0.81 ADORA2A (0.67) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9325950 0.81 ADORA2A (0.76) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL21937216 0.81 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5416151 0.81 ADORA2A (0.66) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9329196 0.80 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL9327337 0.80 ADORA2A (0.69) ADORA2AADORA1ADORA3ADORA2BCSNK1D
SCHEMBL5418348 0.80 ADORA2A (0.64) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL5411130 0.79 ADORA2A (0.63) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed