Bromide

Bromide

SCHEMBL9327702

Br.Cl.O=C(NOCC(O)CN1CCCCC1)c1ccccc1

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 15/20 0.58
MAPK1 P28482 1/20 0.56
CYP2D6 P10635 2/20 0.54
TSHR P16473 1/20 0.54
HIF1A Q16665 1/20 0.54
KDM4E B2RXH2 1/20 0.52
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9329212 0.99 ABCB1 (0.59) ABCB1MAPK1CYP2D6TSHRHIF1A
Hydrochloric Acid SCHEMBL7226297 0.99 ABCB1 (0.59) ABCB1MAPK1CYP2D6TSHRHIF1A
SCHEMBL3073558 0.97 ABCB1 (0.60) ABCB1MAPK1CYP2D6TSHRHIF1A
Hydrochloric Acid SCHEMBL9327623 0.85 ALDH1A1 (0.47) ABCB1MAPK1CYP2D6CYP2C19
SCHEMBL25847563 0.85 ABCB1 (0.50) ABCB1MAPK1CYP2D6TSHRHIF1A
Hydrochloric Acid SCHEMBL28351303 0.85 PRMT5 (0.48) ABCB1MAPK1CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL28996182 0.83 ABCB1 (0.47) ABCB1MAPK1CYP2D6TSHRHIF1A
SCHEMBL5698929 0.82 ABCB1 (0.57) ABCB1MAPK1CYP2D6TSHRHIF1A
Hydrochloric Acid SCHEMBL9329853 0.82 ABCB1 (0.53) ABCB1CYP2D6CYP2C19
SCHEMBL3572645 0.82 ABCB1 (0.47) ABCB1MAPK1CYP2D6TSHRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5328906-A 0-(3-amino-2-hydroxypropyl)-hydroximic acid halides and process for preparing the same BIOREX KUTATO-FEJLESZTO KFT (HU) 1994-07-12 US disclosed
US-5296606-A O-(3-amino-2-hydroxypropyl)-hydroximic acid halides and process for preparing the same BIOREX KUTATO-FEJLESZTO KFT (HU) 1994-03-22 US disclosed
EP-0417210-B1 NOVEL O-(3-AMINO-2-HYDROXYPROPYL)-HYDROXIMIC ACID HALIDES AND PROCESS FOR PREPARING THE SAME BIOREX KUTATO FEJLESZTOE KFT (HU) 1994-03-09 EP disclosed
US-5147879-A O-(3-AMINO-2-HYDROXYPROPYL)-HYDROXIMIC ACID HALIDES AND PROCESS FOR PREPARING THE SAME BIOREX KUTATO-FEJLESZTO KFT (HU) 1992-09-15 US disclosed
WO-1990004584-A1 NOVEL O-(3-AMINO-2-HYDROXYPROPYL)-HYDROXIMIC ACID HALIDES AND PROCESS FOR PREPARING THE SAME BIOREX KUTATÓ FEJLESZTO^' KFT. (HU) 1990-05-03 WO disclosed