SCHEMBL932814

SCHEMBL932814

O=C(NC1=NC[C@H]2COC[C@]2(c2cc(F)cc(NC(=O)c3ccc(F)cn3)c2)S1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 16/20 0.46
BACE2 Q9Y5Z0 8/20 0.43
P4HTM Q9NXG6 3/20 0.39
HDAC3 O15379 1/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932395 0.87 BACE1 (0.55) BACE1BACE2
SCHEMBL932924 0.85 BACE1 (0.56) BACE1BACE2
Hydrochloric Acid SCHEMBL932889 0.84 BACE1 (0.55) BACE1BACE2
SCHEMBL970337 0.81 BACE1 (0.56) BACE1BACE2
SCHEMBL3696178 0.78 BACE1 (0.58) BACE1BACE2
SCHEMBL16056061 0.78 BACE1 (0.44) BACE1P4HTMHDAC3NCOR2
SCHEMBL16027180 0.77 BACE1 (0.47) BACE1BACE2
SCHEMBL16056613 0.75 BACE1 (0.58) BACE1BACE2
SCHEMBL933505 0.75 CYP1A2 (0.36) BACE1HDAC3NCOR2
SCHEMBL18192863 0.75 BACE1 (0.58) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-A1 BACE INHIBITORS Eli Lilly and Company (US) 2012-05-16 EP disclosed
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed