SCHEMBL932924

SCHEMBL932924

NC1=NC[C@H]2COC[C@]2(c2cc(F)cc(NC(=O)c3ccc(F)cn3)c2)S1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.56
BACE2 Q9Y5Z0 8/20 0.52
CTSD P07339 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL932889 0.99 BACE1 (0.55) BACE1BACE2CTSD
SCHEMBL932340 0.85 BACE1 (0.67) BACE1BACE2CTSD
SCHEMBL934283 0.85 BACE1 (0.67) BACE1BACE2CTSD
SCHEMBL932814 0.85 BACE1 (0.46) BACE1BACE2
Hydrochloric Acid SCHEMBL932077 0.84 BACE1 (0.66) BACE1BACE2CTSD
SCHEMBL966237 0.80 BACE1 (0.74) BACE1BACE2CTSD
Hydrochloric Acid SCHEMBL968228 0.79 BACE1 (0.73) BACE1BACE2CTSD
SCHEMBL3696178 0.73 BACE1 (0.58) BACE1BACE2CTSD
SCHEMBL16056555 0.72 BACE1 (0.69) BACE1BACE2CTSD
SCHEMBL6878650 0.72 BACE1 (0.75) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-A1 BACE INHIBITORS Eli Lilly and Company (US) 2012-05-16 EP disclosed
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed