SCHEMBL9328756

SCHEMBL9328756

O=C(O)Cc1ccc2c(c1)NCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
MAPT P10636 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
RGS12 O14924 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
APEX1 P27695 1/20 0.44
THPO P40225 1/20 0.44
BLM P54132 1/20 0.44
GNAI1 P63096 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3091261 0.90 PPARG (0.49) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL9325697 0.87 DRD2 (0.51) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL8003028 0.85 PPARG (0.42) KDM4EALDH1A1SMN1; SMN2ACHECA2
SCHEMBL11977139 0.81 GFER (0.47) MAPTHPGDALDH1A1GAATSHR
SCHEMBL28404333 0.81 KDM4E (0.49) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL7426434 0.79 PPARG (0.38) ALDH1A1SMN1; SMN2ACHEPPARGPPARD
SCHEMBL7600296 0.79 DRD2 (0.44) MAPTALDH1A1SMN1; SMN2ACHEPPARG
Phenylacetic Acid SCHEMBL27898390 0.79 AKR1B1 (0.55) ALDH1A1RXRARXRBRXRGLMNA
SCHEMBL5778832 0.78 KDM4E (0.60) KDM4EMAPTHPGDHSD17B10ALDH1A1
SCHEMBL13234685 0.78 CA9 (0.53) KDM4EMAPTHPGDHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1759095-A N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARM INC (US) 2006-04-12 CN disclosed
CN-1204121-C 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2005-06-01 CN disclosed
CN-1253547-A 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2000-05-17 CN disclosed
US-5288749-A Treating central nervous system or cardiovascular disorders ABBOTT LABORATORIES (US) 1994-02-22 US disclosed